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University of Minnesota
43rd Annual MIKI Meeting
Friday, June 3rd, 2005  

3:00 - 6:30 p.m.

Conference Registration at Days Inn University

6:30 - 7:15 p.m.

Welcome Reception, Cash Bar and Student Mixer at McNamara

7:15 p.m.

Buffet Dinner
Saturday, June 4th, 2005

7:00 - 8:45 a.m.

Continental Breakfest, Days Inn University

9:15 a.m.

(Room 3-120 MCB) Cory Kending, Presiding
  Opening Remarks and Welcome
Session I
  (Room 3-120 MCB) John Goodell, Presiding
   

9:30 - 9:50 a.m.

4’-Fluoro Substitution of Desmethylated Arzoxifene Blocks
Quinoid Formation While Maintaining Antiestrogenic Activity
Hong Liu, Gregory R.J. Thatcher, and Judy L. Bolton*
University of Illinois at Chicago

9:50 - 10:10 a.m.

Design and Synthesis of Type-VIa b-Turn Mimics of Prolyl- Xaa-Prolinamide
Ashish P. Vartak and Rodney L. Johnson*
University of Minnesota

10:10 - 10:30 a.m.

The Design, Synthesis, and Biological Evaluation of HSP90 Inhibitors
Gang Shen and Brian S. J. Blagg*
University of Kansas

10:30 a.m.

Break, Coffee and Pasteries provided, 3-120 MCB
Session II

 

 (Room 3-120 MCB) Upendra Argrikar, Presiding

11:00 -12:00 a.m.

 KEYNOTE ADDRESS
Dr. Christopher A. Lipinski, Adjunct Senior Research Fellow,
Groton Laboratories, Pfizer Global Research and Development
   

12:00 a.m.

Lunch 3-120 MCB
Poster Preparation, BSBE 2nd Floor
Session III
  (Room 3-120 MCB) Terry Steele, Presiding
   

1:30 - 1:50 p.m.

Synthetic Studies Toward the Construction of the cis-Decalin Portion of Superstolides A and B. Application of a Sequential Double Michael Reaction and an Anionic Oxy-Cope Rearrangement
Zhengmao Hua, Wensheng Yu, Mei Su, and Zhendong Jin*
University of Iowa

1:50 - 2:10 p.m.

Histidine Triad Nucleotide Binding Proteins (HINT) are Nucleoside
Phosphoramidases and Potential Regulators of Protein Nucleotidylation
Tsui-Fen Chou and Carston R. Wagner
University of Minnesota

2:10 - 2:30 p.m.

Synthesis and Reactions of Twisted Amides
Lei Yao, Aaron D. Wrobleski, Jennifer E. Golden, Jeffrey Aubé *
University of Kansas

2:30 - 2:50 p.m.

Structural Basis for Tumor Pyruvate Kinase M2 Allosteric Regulation and Catalysis
Jill D. Dombrauckas, Bernard D. Santarsiero, and Andrew D.Mesecar
University of Illinois at Chicago
Session IV
  (BSBE 2nd Floor) Jaeson Steele, Presiding

3:00 - 5:00 p.m.

Poster Presentation and Refreshments in BSBE 2nd Floor

3:00 - 5:00 p.m.

Interviews
Saturday Night Banquet  

7:00 - 7:45 p.m.

Cash Bar: Coffman Memorial Union - Great Hall, UMN

7:45 p.m.

Banquet: Coffman Memorial Union - Great Hall, UMN
Sunday, June 5th, 2005  

Check Out

Days Inn University

7:00 - 8:35 a.m.

Continental Breakfest, Days Inn University
Session V
  (Room 3-120 MCB) Annie Nguyen, Presiding
   

8:40 - 9:00 a.m.

Evaluation of the Antinociceptive Activity of Herkinorin and Salvinorin A in a Rodent Model of Nociception
Kevin J. Tidgewell, Wayne W. Harding, Christina M. Dersch, Richard B. Rothman, Thomas E. Prisinzano*
University of Iowa

9:00 - 9:20 a.m.

Novel Taxol Analogs for Brain Delivery
Haibo Ge and Gunda I. Georg*
University of Kansas

9:20 - 9:40 a.m.

Evaluation of Polyethyleneimine-Dextran Block Polymers for use as Non-Viral Vectors in Gene Therapy
Terry W.J. Steele, W.T. Shier*
University of Minnesota

9:40 - 10:00 a.m.

 Mapping Potential New Sites for Antibiotic Action in the Ribosome
Aymen S Yassin and Alexander S Mankin*.
University of Illinois at Chicago

10:00-10:30 a.m.

Break, Coffee and Pastries, 3-120 MCB
Session VI
 

(Room 3-120 MCB) Cory Kending, Presiding

   

10:30 - 10:50 a.m.

Progress Towards the Synthesis of Tubulysin D
Jaeson C. Steele, Venkat Lakshmanan, Courtney C. Aldrich, and Robert A. Fecik*.
University of Minnesota

10:50 - 11:10 a.m.

Oxidative Metabolism of the Serm, Raloxifene Leads to Protein Covalent Modification
Ju Liu, Qian Li, , Xiaofeng Yang, Minsun Chang, Richard B. van Breemen, Gregory R. J. Thatcher, and Judy L. Bolton
University of Illinois at Chicago

11:10 - 11:30 a.m.

 Preparation of Thermally Activatable Phosphoramidate Diesters for Intracellular Pronucleotide Delivery
Dan P. Drontle, Dr. A. O. Akanni, Dr. Y. J. Abul-Hajj, and Dr. C. R. Wagner*
University of Minnesota
   

11:30 a.m.

Adjournment Faculty Meeting

12:15 p.m.

Pick up Boxed Lunch at 3-120 MCB

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